Experiment 348595
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | WANG,BQ: PANG,ZG: WANG,CY: YI,H:. (1995). STUDY ON PHARMACOKINETIC PARAMETERS OF ANDROGRAPHOLIDE IN RABBIT PLASMA BY CHEMILUMINESCENCE.. 12(1) |
| Amount utilized | |
| Compound isolated | |
| Disease | THE BLOOD CONCENTRATION OF ANDROGRAPHOLIDE WAS MONITORED BY A HIGHLY SENSITIVE ORG. COUPLED CHEMILUMINESCENCE TECHNIQUE AND A SERIES OF PHARMACOKINETIC PARAMETERS WERE OBTAINED. THE RESULTS SUGGEST THAT ANDROGRAPHOLIDE CAN RAPIDLY REACH PEAK CONCENTRATION. THE HALF-LIFE OF ITS ELIMINATION IS LONG AND THE BIOAVAILABILITY IS HIGH. THE MAIN PHARMACOKINETIC PARAMETERS ARE: KA- 1.34/H + 0.08, K1.2=0.336/H+0.01, K2.1-0.633/H+ 0.06, T0.5(A)=10.692 H + 0.07, T(A)=12.12H + 1.9, AUC=501.09 MG.H/ML+ 9.8. |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RABBIT |
| Dose expression | DOSE |