Experiment 349616

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationOARTENSI,G: GLADSTEIN,J: VALLI,H: TESONE,PA:. (1997). A COMAPRATIVE STUDY OF POLICOSANOL VERSUS SIMVASTATIN IN ELDERLY PATIENTS WITH HYPERCHOLESTEROLEMIA.. 58(6)
Amount utilized
Compound isolated
DiseaseFIFTY-THREE ELDERLY PATIENTS (60 TO 77 YEARS OF AGE) WITH PRIMARY HYPERCHOLESTEROLEMIA (TOTAL SERUM CHOLESTEROL >240 MG/DL) WERE ENROLLED IN A RANDOMIZED, DOUBLE-MASKED, PARALLEL-GROUP, COMPARATIVE STUDY OF POLICOSANOL, AND SIMVASTATIN. BEFORE RANDOMIZATION, ALL PATIENTS WERE ADVISED TO FOLLOW A STANDARD CHOLESTEROL-LOWERING DIET FOR 6 WEEKS. PATIENTS WERE RANDOMIZED TO RECEIVE ETHER POLICOSANOL OR SIMVASTATIN, BOTH AT DOSES OF 10 MG/D FOR 8 WEEKS. WITH POLICOSANOL, TOTAL CHOLESTEROL, LOW-DENSITY LIPOPROTEIN CHOLESTEROL (LDL-C), AND TRIGLYCERIDES WERE SIGNIFICANTLY REDUCED 14.7%, 17.9%, AND 13.8%, RESPECTIVELY. SIMVASTATIN SIGNIFICANTLY LOWERED TOTAL CHOLESTEROL 15.2%, LDL-C 19.8%, AND TRIGLYCERIDES 8.7%. NEITHER POLICOSANOL NOR SIMVASATIN SIGNIFICANTLY CHANGED HIGH-DENSITY LIPOPROTEIN CHOLESTEROL (HDL-C) LEVELS. TOTAL CHOLESTEROL:HDL-C AND LDL-C:HDL-C RATIOS WERE SIGNIFICANTLY LOWERED BY BOTH THERAPIES. THE EFFECTS OF BOTH DRUGS ON LIPID PROFILE VARIABLES WERE STATISTICALLY SIMILAR. BOTH DRUGS WERE WELL TOLERATED.
Dose amount10.0 MG
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitKG
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES