Experiment 362520

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismCitrus paradisi (RUTACEAE)
CitationFELDMAN,EB:. (1997). HOW GRAPEFRUIT JUICE POTENTIATES DRUG BIOAVAILABILITY.. 55(11)
Amount utilized
Compound isolated
DiseaseLIKELY ACCELERATES BREAKDOWN OF CYTOCHROME P3A4 OR/AND TRANSLATION OF MRNA FOR SAME, THERAPY INCREASING BIOAVAILABILITY OF DRUGS METABOLIZED BY THIS CYTOCHROME IN COLONIC BRUSH BORDER.
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Dose expressionDOSE
ExtractJUICE