Experiment 372320

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeINTRAVESICULAR
OrganismEmpty organism
CitationDASGUPTA,P: CHANDIRAMANI,V: PARKINSON,MC: BECKETT,A: FOWLER,CJ:. (1998). TREATING THE HUMAN BLADDER WITH CAPSAICIN: IS IT SAFE?. 33(1)
Amount utilized
Compound isolated
DiseaseBETWEEN 1991 AND 1996, 20 PTS (9 MALES, 11 FEMALES; MEAN AGE 52.5 YRS. RANGE 40-70 YRS) WITH INTRACTABLE DETRUSOR HYUPERREFLEXIA HAVE HAD REPEATED INSTILLATIONS OF INTRAVESICAL CAPSAICIN (1-2 MMOL/L). THE NUMBER OF TREATMENTS PER PTS VARIED BETWEEN 1 AND 17 (TOTAL-82; AVERAGE 6/PT). THE SURVEILLANCE PROGRAMME INVOLVED REPEATED FLEXIBLE CYSTOSCOPY AND BLADDER BIOPSIES BEFORE AND AFTER CAPSAICIN. CRYOSTAT SECTIONS WERE STRAINED WITH HAEMTOXYLIN-EOSIN AND EXAMINED BY LIGHT MICROSCOPY. NONE OF THE BLADDER BIOPSIES HAVE SHOWN METAPLASIA, DYSPLASIA, FLAT CARCINOMA IN SITU, PAPILLARY OR SOLID INVASIVE CANCER. NO PRE-MALIGNANT OF MALIGNANT CHANGE HAS BEEN FOUND IN BIOPSIES OF PATIENTS WHO HAD REPEATED CAPSAICIN INSTILLATIONS FOR UP TO 5 YRS.
Dose amount0.3 GM
Number1
Qualitative resultINACTIVE
AnimalHUMAN ADULT
Per unitLITER
Dose expressionDOSE
GenderGIVEN TO BOTH SEXES