Experiment 374157
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | DAHLSTROM,B: MELLSTRAND,T: LOFDAHL,CG: JOHANSSON,M:. (1982). PHARMAKOKINETIC PROPERTIES OF NOSCAPINE.. 22() |
| Amount utilized | |
| Compound isolated | |
| Disease | NOSCAPINE WAS ADMINISTERED TO FIVE HEALTHY VOLUNTEERS IN A RANDOMIZED CROSSOVER DESIGN, AS AN INTRAVENOUS INFUSION OF 66 MG, AND AS AN ORAL 150 MG DOSE OF EITHER RAPIDLY DISSOLVING TABLETS OR A TABLET CONTAINING ION EXCHANGE RESIN-BOUND NOSCAPINE. AFTER I.V. ADMINISTRATION, THE DISPOSITION OF NOSCAPINE WAS BI-EXPONTENTIAL WITH AN ELIMINATION HALF-LIFE OF 2.6 H; THE TOTAL PLASMA CLEARANCE WAS 22 M./MIN/KG AND THE VOLUME OF DISTRIBUTION (VD AREA) WAS 4.7 1/KG. |
| Dose amount | 66.0 MG |
| Number | 1 |
| Qualitative result | . |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |
| Gender | GIVEN TO BOTH SEXES |