Experiment 375562

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismEmpty organism
CitationSHOBA,G: JOY,D: JOSEPH,T: MAJEED,M: RAJENDRAN,R: SRINIVAS,PSSR:. (1998). INFLUENCE OF PIPERINE ON THE PHARMACOKINETICS OF CURCUMIN IN ANIMALS AND HUMAN VOLUNTEERS.. 64(4)
Amount utilized
Compound isolated
DiseaseA DOSE OF 2 G CURCUMIN ALONE, SERUM LEVELS WERE EITHER UNDETECTABLE OR VERY LOW. CONCOMITANT ADMINISTRATION OF PIPERINE 20 MG PRODUCED MUCH HIGHER CONCENTRATIONS FROM 0.25 TO 1 HOUR POST DRUG (P<0.01 AT 0.25 AND 0.5 HOUR; P<0.001 AT 1 HOUR), THE INCREASE IN BIOAVAILABILITY WAS 2000%. THE STUDY SHOWS THAT IN THE DOSAGES USED, PIPERINE ENHANCES THE SERUM CONCENTRATION, EXTENT OF ABSORPTION AND BIOAVAILABILITY OF CURCUMIN IN HUMANS WITH NO ADVERSE EFFECTS.
Dose amount2.0 GM
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitKG
Dose expressionDOSE
GenderMALE