Experiment 417763

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationMINISCALCO,A: LUNDAHL,J: REGARDH,CG: EDGAR,B: ERIKSSON,UG:. (1992). INHIBITION OF DIHYDROPYRIDINE METABOLISM IN RAT AND HUMAN LIVER MICROSOMES BY FLAVONOIDS FOUND IN GRAPEFRUIT JUICE.. 261(2)
Amount utilized
Compound isolated
DiseaseTHE SUBTYPE III4A OF GIVEN ENZYME IS INHIBITED, PREVENTING THE OXIDATION OF DIHYDROPYRIDINES, THEREBY INHIBITING THE METABOLISM OF (R)-FELODIPINE.
Dose amount100.0 MICROMOLS
Number4
Qualitative resultACTIVE
AnimalRAT
Dose expressionCONC USED