Experiment 426816
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Streptomyces species (STREPTOMYCETACEAE) |
| Citation | KUWAHARA,T: KUDOH,T: NAGASE,H: TAKAMIYA,M: NAKANO,A: OHTSUKA,T: YOSHIZAKI,H: ARISAWA,M:. (1992). TETRONOTHIODIN, A NOVEL CCK-B RECEPTOR LIGAND, ANTAGONIZES CHOLECYSTOKININ-INDUCED CA2+ MOBILIZATION IN A PITUITARY CELL LINE.. 221(1) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND INHIBITED BINDING OF LABELLED CCK-8 TO CCK-B RECEPTORS. IT IS 20,000 LESS EFFECTIVE AS CCK-A RECEPTOR ANTAGONIST. |
| Dose amount | 3.6 NANOMOLS |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Dose expression | IC50 |