Experiment 428494

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationSAGARA,Y: FERNANDEZ-BELDA,F: DE MEIS,L: INESI,G:. (1992). CHARACTERIZATION OF THE INHIBITION OF INTRACELLULAR CA2+ TRANSPORT ATPASES BY THAPSIGARGIN.. 267(18)
Amount utilized
Compound isolated
DiseaseCOMPOUND IRREVERSIBLY INHIBITS ENZYME BY BINDING TO STATE ACHIEVED DURING TURNOVER OF ENZYME IN ABSENCE OF ATP, CA2+ INHIBITS BINDING OF COMPOUND.
Dose amount2.0 NANOMOLS
Number1
Qualitative resultACTIVE
Per unitPER MG PROTEIN
Dose expressionCONC USED