Experiment 428496

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationKIRBY,MS: SAGARA,Y: GAA,S: INESI,G: LEDERER,WJ: ROGERS,TB:. (1992). THAPSIGARGIN INHIBITS CONTRACTION AND CA2+ TRANSIENT IN CARDIAC CELLS BY SPECIFIC INHIBITION OF THE SARCOPLASMIC RETICULUM CA2+ PUMP.. 267(18)
Amount utilized
Compound isolated
DiseaseINTRACELLULAR CA2+ CONC. TRANSIENT INCREASE IS INHIBITED. CA2+-INDUCED CA2+ RELEASE IS NOT AFFECTED WHILE CA-ATPASE ACT IS INHIBITED.
Dose amount100.0 NANOMOLS
Number2
Qualitative resultACTIVE
AnimalRAT
Dose expressionCONC USED