Experiment 431918
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | GUSOVSKY,F: PADGETT,WL: CREVELING,CR: DALY,JW:. (1992). INTERACTION OF PUMILIOTOXIN B WITH AN "ALKALOID-BINDING DOMAIN ON THE VOLTAGE-DEPENDENT SODIUM CHANNEL.. 42(6) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND ACTIVITES VOLTAGE-DEPENDENT CHANNELS. EFFECT POTENTIATED BY ALPHA AND BETA SCORPION TOXINS AND BREVETOXIN WHICH IS NOT TRUE OF VERATRIDINE. UNLIKE ACONITINE, COMPOUND DOES NOT INHIBIT BINDING OF BATRACHOTOXININ-A BENZOATE. COMPOUND'S EFFECTS INHIBITED BY BOTH TYPE I AND II PYRETHROIDS, AS IS THE EFFECT OF ACONITINE. |
| Dose amount | 100.0 MICROMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | GUINEA PIG |
| Dose expression | CONC USED |