Experiment 440211
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | BOCCHIO,F: KALF-HANSEN,S: DEKERMENDJIAN,K: STERNER,O: WITT,R:. (1992). THE INHIBITORY EFFECT OF SESQUITERPENOID UNSATURATED DIALDEHYDES ON THE DOPAMINE D1 RECEPTOR, A QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIPS STUDY.. 33(45) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND INHIBITED BINDING OF TRITIATED SCH 23390 ((R)-(+)-8-CHLORO-2, 3, 4, 5-TETRAHYDRO-3-METHYL-5-PHENYL-1H-3-BENZAZEPIN-7-OL) TO DOPAMINE-1 RECEPTORS. |
| Dose amount | 0.31 MICROMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Dose expression | IC50 |