Experiment 441069
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | FELIX,JP: KING,VF: SHEVELL,JL: GARCIA,ML: KACZOROWSKI,GJ: BICK,IRC: SLAUGHTER,RS:. (1992). BIS(BENZYLISOQUINOLINE) ANALOGS OF TETRANDRINE BLOCK L-TYPE CALCIUM CHANNELS: EVIDENCE FOR INTERACTION AT THE DILITAZEM-BINDING SITE.. 31(47) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND INHIBITS BINDING OF DILTIAZEM, D-600, FLUSPIRILENE AND NITRENDIPINE. INHIBITION OF DILTIAZEM BINDING CORRELATES WITH CA2+ UPTAKE INHIBITION. IC-50 VALUE GIVEN FOR DILTIAZEM BINDING AT 37C. |
| Dose amount | 0.84 MICROMOLS |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | PIG |
| Dose expression | IC50 |