Experiment 442350
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | LINGHAM,RB: HSU,A: SILVERMAN,KC: BILLS,GF: DOMBROWSKI,A: GOLDMAN,ME: DARKE,PL: HUANG,L: KOCH,G: ONDEYKA,JG: GOETZ,MA:. (1992). L-696,474, A NOVEL CYTOCHALASIN AS AN INHIBITOR OF HIV-1 PROTEASE III. BIOLOGICAL ACTIVITY.. 45(5) |
| Amount utilized | |
| Compound isolated | |
| Disease | HIV-1 PROTEASE ACTIVITY INHIBITION WAS COMPETATIVE WITH RESPECT TO THE SUBSTRATE. |
| Dose amount | 3.0 MICROMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Dose expression | IC50 |