Experiment 446789

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationKASAI,M: KAWASAKI,T:. (1993). EFFECTS OF RYANODINE ON PERMEABILITY OF CHOLINE AND GLUCOSE THROUGH CALCIUM CHANNELS IN SARCOPLASMIC RETICULUM VESICLES.. 113(3)
Amount utilized
Compound isolated
DiseaseCMPD LOCKED CA-INDUCED CA. CHANNEL OPEN. CHOLINE BECAME PERMEABLE EVEN IN ABSENCE OF CA. SIMILARY, GLUCOSE BECAME PERMEABLE IN ABSENCE OF KCL. ACTIVATORS OF CHANNEL SUCH AS ATP AND CAFFEINE DID NOT ENHANCE EFFECT WHILE INHIBITORS SUCH AS MG AND RUTHENIUM RED INHIBITED EFFECT. HIGHER CONC. OF CMPD (100 MICROMOLAR) CLOSED CHANNEL.
Dose amount10.0 MICROMOLS
Number1
Qualitative resultACTIVE
Dose expressionCONC USED