Experiment 449518

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationWONG,S: MOK,W: PHANEUF,S: KATZ,S: SALARI,H:. (1993). FORSKOLIN INHIBITS PLATELET-ACTIVATING FACTOR BINDING TO PLATELET RECEPTORS INDEPENDENTLY OF ADENYLYL CYCLASE ACTIVATION.. 245(1)
Amount utilized
Compound isolated
DiseaseEXPOSURE TO COMPOUND FOR 2 MIN DECREASED MUNBER OF PAF RECEPTORS AVAILABLE. ANALOGUES OF CAMP DID NOT HAVE EFFECT. NEITHER DID EXPOSURE TO PGE2 WHICH RESULTED IN INCREASED CAMP LEVELS. EFFECT WAS ADDITIVE TO THAT OF GTP-GAMMA S. PHOSPHOKINASE INHIBITORS A3 AND STAUROSPORINE DID NOT HAVE GIVEN EFFECT.
Dose amount50.0 MICROMOLS
Number2
Qualitative resultACTIVE
AnimalRABBIT
Dose expressionCONC USED