Experiment 451843
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | CHEN,G: RAMACHANDRAN,C: KRISHAN,A:. (1993). THALIBLASTINE, A PLANT ALKALOID, CIRCUMVENTS MULTIDRUG RESISTANCE BY DIRECT BINDING TO P-GLYCOPROTEIN.. 53(11) |
| Amount utilized | |
| Compound isolated | |
| Disease | 1 HOUR EXPOSURE TO COMPOUND REDUCED ID-50 OF ADRIAMYCIN FROM 10.8 TO 1.4 MICROMOLAR. 24 HOURS EXPOSURE REDUCED ID-50 FROM 3.5 TO 0.07 MICROMOLAR. ADRIAMYCIN RETENTION ENHANCED. PHOTO LABELING OF P-GLYCOPROTEIN WITH AZIDOPINE INHIBITED. |
| Dose amount | 2.0 MICROMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | CONC USED |