Experiment 455817

Details

PropertyValue
Pharmacology
OrganismSetosphaeria khartoumensis (PYRENOPHORACEAE)
CitationHASUMI,K: TACHIKAWA,K: SAKAI,K: MURAKAWA,S: YOSHIKAWA,N: KUMAZAWA,S: ENDO,A:. (1993). COMPETITIVE INHIBITION OF SQUALENE SYNTHETASE BY SQUALESTATIN I.. 46(4)
Amount utilized
Compound isolated
DiseaseTHE INHIBITION WAS 79%. THE REACTION WAS MEASRUED BY FORMATION FROM [3H] PSPP IN THE PRESENCE OF NADPH. THIS WAS 2ND PARTIAL REACTION.
Dose amount33.4 NANOMOLS
Number4
Qualitative resultSTRONG ACTIVITY
Dose expressionDOSE