Experiment 470571

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationHERBERT,JM: SAVI,P: LAPLACE,MC: DUMAS,A: DOL,F:. (1993). CHELERYTHRINE, A SELECTIVE PROTEIN KINASE C INHIBITOR, COUNTERACTS PYROGEN-INDUCED EXPRESSION OF TISSUE FACTOR WITHOUT EFFECT ON THROMBOMODULIN DOWN-REGULATION IN ENDOTHELIAL CELLS.. 71(6)
Amount utilized
Compound isolated
DiseaseVS.IL-1BETA INDUCED UPREGULATION OF TISSUE FACTOR. CONCOMITANT DOWN REGULATIN OF THROMBOMODULIN NOT ALTERED BY CMPD.
Dose amount6.6 MICROMOLS
Number1
Qualitative resultACTIVE
AnimalBULL
Dose expressionIC50