Experiment 481538
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | SCOTT,DO: BINDRA,DS: STELLA,VJ:. (1993). PLASMA PHARMACOKINETICS OF THE LACTONE AND CARBOXYLATE FORMS OF 20(S)-CAMPTOTHECIN IN ANESTHETIZED RATS.. 10(10) |
| Amount utilized | |
| Compound isolated | |
| Disease | INITIAL PLASMA CONCENTRATIONS OF THE LACTONE WERE SIGNIFICANTLY HIGHER AFTER DOSING WITH THE LACTONE OF CPT THAN AFTER DOSING WITH ITS SODIUM SALT. AFTER 90 MIN, CONCENTRATION OF THE LACTONE APPEARS INDEPENDENT OF THE FORM ADMINISTERED. THE SAME APPEARS TO BE TRUE FOR THE CARBOXYLATE OF CPT. |
| Dose amount | 1.0 MG |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Per unit | KG |
| Dose expression | DOSE |