Experiment 481820

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeINTRACRANIAL
OrganismEmpty organism
CitationALBUQUERQUE,MLC: KURTH,CD:. (1993). COCAINE CONSTRICTS IMMATURE CEREBRAL ARTERIOLES BY A LOCAL ANESTHETIC MECHANISM.. 249(2)
Amount utilized
Compound isolated
DiseaseCOMPOUND IN CONC. OF 0.1 MICROMOLAR-1.0 MILLIMOLAR CAUSED DOSE-DEPENDENT CONSTRICTION OF ARTERIOLES VISUALIZED THROUGH CLOSED CRANIAL WINDOW PREPARATION. PHENTOLAMINE DID NOT INHIBIT EFFECT WHILE TETRODOTOXIN, CHARYBDOTOXIN, QUINACRINE OR INDOMETHACINE DID. LIDOCAINE HAD SIMILAR EFFECT ON ARTERIOLES AS COMPOUND.
Dose amountVAR
Number1
Qualitative resultACTIVE
AnimalPIG
Dose expressionDOSE