Experiment 483535

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismStreptomyces neyagawaensis (STREPTOMYCETACEAE)
CitationSATOH,T: YAMASHITA,Y: KAMIYAMA,T: WATANABE,J: STEINER,B: HADVARY,P: ARISAWA,M:. (1993). TETRAFIBRICIN: A-NONEPTIDIC FIBRINOGEN RECEPTOR INHIBITOR FROM STREPTOMYCES NEYAGAWAENSIS (I) ITS GPIIB/IIIA BLOCKAGE ON SOLID PHASE BINDING ASSAY.. 72(5)
Amount utilized
Compound isolated
DiseaseCOMPOUND INHIBITS BINDING OF FIBRINOGEN, FIBRONECTIN AND VON WILLEBRAND FACTOR TO GPIIB/IIIA.
Dose amount46.0 NANOMOLS
Number2
Qualitative resultACTIVE
Dose expressionIC50