Experiment 489083
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | PIEK,T: HUE,B: LE CORRONE,H: MANTEL,P: GOBBO,M: ROCCHI,R:. (1993). PRESYNAPTIC BLOCK OF TRANSMISSION IN THE INSECT CNS BY MONO- AND DIGALACTOSYL ANALOGS OF VESPULAKININ 1, A WASP (PARAVESPULA MACULIFRONS) VENOM NEUROTOXIN.. 105(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | TWO EFFECTS WERE OBSERVED; THEY ARE, A DIRECT AND REVERSIBLE BLOCK OF EXCITATORY NICOTINIC TRANSMISSION WITH A CONCURRENT ACTIVATION OF THE INHIBITORY GABAERGIC SYSTEM, AND A DELAYED IRREVERSIBLE BLOCK OF THE TRANSMISSION. FOR THIS STUDY, MAMMALIAN SMOOTH MUSCLE AND SYNAPTIC TRANSMISSION FROM THE COCKROACH CERCAL NERVES TO A GIANT INTERNEURON. |
| Number | 1 |
| Qualitative result | ACTIVE |
| Dose expression | CONC USED |