Experiment 489507

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationHASHIMOTO,Y: WATANABE,T: KINOSHITA,M: TSUKAMOTO,K: TOGO,M: HORIE,Y: MATSUDA,Y: KUROKAWA,K:. (1993). CA2+ ENTRY PATHWAYS ACTIVATED BY THE TUMOR PROMOTER THAPSIGARGIN IN HUMAN PLATELETS.. 1220(1)
Amount utilized
Compound isolated
DiseaseWORTMANNIN PARTIALLY ANTAGONIZED EFFECT. THIS CMPD AND THE TXA-S RECEPTOR ANTAGONIST S-145 INHIBITED THAPSIGARIN INDUCED PHOSPHORYLATION OF MYOSIN LIGHT CHAIN KINASE AND A PROTEIN KINASE C SUBSTRATE, 47-KDA PROTEIN.
Dose amount0.2 MICROMOLS
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Dose expressionCONC USED