Experiment 489856
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | SHOSHAN-BARMATZ,Y: ZCHUT,S:. (1993). THE INTERACTION OF LOCAL ANESTHETICS WITH THE RYANODINE RECEPTOR OF THE SARCOPLASMIC RETICULUM.. 133(2) |
| Amount utilized | |
| Compound isolated | |
| Disease | TETRACAINE AND DIBUCAINE INHIBIT THE BINDING OF RYANODINE WITH AN IC50 OF 0.12 AND 0.25 MM RESP.LIDOCAINE, ITS ANALOG QX-314 AND PRILOCAINE STIMULATE THE BINDING UP TO FOURFOLD WITH HALF-MAXIMAL STIMULATION OCCURRING WITH ABOUT 2MM OF DRUGS. |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | CONC USED |