Experiment 490272

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationWALLE,T: KUMAR,GN: MC MILLAN,JM: THORNBURG,KR: WALLE,UK:. (1993). TAXOL METABOLISM IN RAT HEPATOCYTES.. 46(9)
Amount utilized
Compound isolated
DiseaseMETABOLISM OF TAXOL YIELDED 2 METABOLITIES M-1 AND M-2, WITH K-M VALUES OF 68 AND 61 MICROMOLS. METABOLISM WAS INHIBITED BY VERAPAMIL AND MIDAZOLAM AT IC-50 DOSES OF 100 AND 25 MICROMOLS RESPECTIVELY.
Dose amount30.0 MICROMOLS
Number1
Qualitative result.
AnimalCELL CULTURE
Dose expressionCONC USED