Experiment 492259

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismDaucus carota (APIACEAE)
CitationYANG,WN: BOSS,W:. (1994). REGULATION OF PHOSPHATIDYLINOSITOL 4-KINASE BY THE PROTEIN ACTIVATOR PIK-A49.. 269(5)
Amount utilized
Compound isolated
DiseasePIK-A49 DECREASED THE KM OF PI 4-KINASE FOR ATP FROM 0.40 TO 0.19 NM. GTP AND GDP INHIBITED THE ACTIVATION OF PI 4-KINASE BY PIK-A49. PHOSPHORYLATION OF PIK-A49 BY A CALCIUM DEPENDENT PROTEIN KINASE ENHANCED ACTIVATION OF PI 4-KINASE.
Dose amount22.0 MCG
Number2
Qualitative resultACTIVE
Per unitML
Dose expressionCONC USED