Experiment 493142

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationIYER,RS: COLES,BF: RANEY,KD: THIER,R: GUENGERICH,FP: HARRIS,TM:. (1994). DNA ADDUCTION BY THE POTENT CARCINOGEN AFLATOXIN B-1: MECHANISTIC STUDIES.. 116(5)
Amount utilized
Compound isolated
DiseaseCOMPOUND METABOLIZED TO EXO- AND ENDO- 8,9-EPOXIDES. EXO COMPOUND UNDERGOES SN2 RXN WITH GUANINE WHILE ENDO FAILS TO FROM ADDUCT WITH GUANINE AND IN FACT IS NOT MUTAGENIC.
Dose amount2.0 MG
Number1
Qualitative resultACTIVE
Per unitML
Dose expressionCONC USED