Experiment 493864
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Dendroaspis angusticeps (ELAPIDAE) |
| Citation | SCHWEITZ,H: HEURTEAUX,C: BOIS,P: MOINIER,D: ROMEY,G: LAZDUNSKI,M:. (1994). CALCICLUDINE, A VENOM PEPTIDE OF THE KUNITZ-TYPE PROTEASE INHIBITOR FAMILY, IS A POTENT BLOCKER OF HIGH-THRESHOLD CA(2+) CHANNELS WITH A HIGH AFFINITY FOR L-TYPE CHANNELS IN CEREBELLAR GRANULE NEURONS.. 91(3) |
| Amount utilized | |
| Compound isolated | |
| Disease | LABELED CMPD BINDS TO OLFACTORY BULB, MOLECULAR LAYER OF DENTATE GYRUS, STRATUM ORIENS OF CA3 FIELD OF HIPPOCAMPAL FORMATION, AND GRANULAR LAYER OF CEREBELLUM. BLOCKS L-SUBTYPE NEURONAL CA(2+) CHANNELS. |
| Dose amount | 5.0 NANOMOLS |
| Number | 2 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Dose expression | CD90 |