Experiment 505616

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeINTRAGASTRIC
OrganismEmpty organism
CitationNAKAMURA,M: IMAOKA,S: MIURA,K: TANAKA,F: MISAWA,S: FUNAE,Y:. (1994). INDUCTION OF CYTOCHROME P450 ISOZYMES IN RAT RENAL MICROSOMES BY CYCLOSPORIN A.. 48(9)
Amount utilized
Compound isolated
DiseaseDOSED DAILY X17 DAYS. EFFECT SEEN ON CYP4A2 BUT NOT ON CYP2C23, CYP3A1 OR CYP4A8. INCREASED LEVELS OF OMEGA-HYDROXYL- AND OMEGA-1-HYDROXY-ARACHIDONATE ARE SEEN, WHICH MAY CONTRIBUTE TO RENAL PATHOLOGY.
Dose amount50.0 MG
Number1
Qualitative resultACTIVE
AnimalRAT
Per unitKG
Dose expressionDOSE