Experiment 506274

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationPOWIS,G: GALLEGOS,A: ABRAHAM,RT: ASHENDEL,CL: ZALKOW,LH: GRINDEY,GB: BONJOUKLIAN,R:. (1994). INCREASED INTRACELLULAR CA2+ SIGNALING CAUSED BY THE ANTITUMOR AGENT HELENALIN AND ITS ANALOGUES.. 34(4)
Amount utilized
Compound isolated
DiseaseHELENALIN AT BETWEEN O.1 AND 10 MICROGRAMS PER MILLILITER CAUSED A 175% INCREASE IN 45 CA2+ UPTAKE. THE SAME CONCENTRATIONS OF HELENALIN CAUSED A 260% INCREASE IN THE INS(1,4,5) P3-DEPENDENT RELEASE OF 45CA2+.
Dose amount0.10 MCG
Number6
Qualitative resultACTIVE
AnimalCELL CULTURE
Per unitML
Dose expressionCONC USED