Experiment 510252
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | LI,Y: KOBAYASHI,H: HASHIMOTO,Y: SHIRAI,R: HIRATA,A: HAYASHI,K: HAMADA,Y: SHIOIRI,T: IWASAKI,S:. (1994). INTERACTION OF MARINE TOXIN DOLASTATIN 10 WITH PORCINE BRAIN TUBULIN: COMPETITIVE INHIBITION OF RHIZOXIN AND PHOMOPSIN A BINDING.. 93(3) |
| Amount utilized | |
| Compound isolated | |
| Disease | DOLASTATIN 10 INHIBITED THE BINDING OF RADIO LABELLED RHIZOXIN TO TUBULIN WITH INHIBITION CONSTANT (KI) OF 7 X 10-8 M. |
| Dose amount | 70.0 NANOMOLS |
| Number | 3 |
| Qualitative result | ACTIVE |
| Dose expression | IC50 |