Experiment 515013

Details

PropertyValue
Pharmacology
OrganismPiper methysticum (PIPERACEAE)
CitationJUSSOFIE,A: SCHMIZ,A: HIEMKE,C:. (1994). KAVAPYRONE ENRICHED EXTRACT FROM PIPER METHYSTICUM AS MODULATOR OF THE GABA BINDING SITE IN DIFFERENT REGIONS OF RAT BRAIN.. 116(4)
Amount utilized
Compound isolated
DiseaseENHANCED BINDING OF LABELED MUSCIMOL BY INCREASING NUMBER OF BINDING SITES. EFFECT SEEN IN HIPPOCAMPUS, AMYGDALA, MEDULLA OBLONGATA, FRONTAL CORTEX AND CEREBELLUM. EFFECT ENHANCED BY PENTOBARBITAL AND 3-ALPHA-HYDROXY-5-ALPHA-PREGNANE-20-ONE.
Dose amount300.0 MICROMOLS
Number1
Qualitative resultACTIVE
AnimalRAT
Dose expressionED50
ExtractCHROMATOGRAPHIC FRACTION