Experiment 515874

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationMAGUIRE,JJ: BACON,CR: FUJIMOTO,M: DAVENPORT,AP:. (1994). MYRICERONE CAFFEOYL ESTER (50-235) IS A NON-PEPTIDE ANTAGONIST SELECTIVE FOR HUMAN ETA RECEPTORS.. 12(6)
Amount utilized
Compound isolated
DiseaseINTERNAL MAMMARY ARTERY USED. COMPETITIVELY INHIBITED ET-1-INDUCED CONSTRICTION. PA2 VALUES GIVEN.
Dose amount6.18 MOL
Number3
Qualitative resultACTIVE
AnimalHUMAN ADULT
Dose expression-LOG(CONC.)