Experiment 516956

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationYAZDANBAKHSH,K: WON,JW: LI,YZ: LAU,LF: CHOI,YW:. (1995). CYCLOSPORIN A BLOCKS APOPTOSIS BY INHIBITING THE DNA BINDING ACTIVITY OF THE TRANSCRIPTION FACTOR NUR77.. 92(2)
Amount utilized
Compound isolated
DiseaseVS.T-CELL RECEPTOR MEDIATED APOPTOSIS OF THYMOCYTES CSA INHIBITS THE TCR-MEDIATEE ACTIVATION OF NUR77 PROTEIN IN T-CELL HYBRIDOMAS BY BLOCKING THE DNA BINDING ACTIVITY OF NUR77 PROTEIN RATHER THAN ITS DE NOV SYNTHESIS. CSA MEDIATES ITS NEGATIVE EFFECTS ON THE NUR77 DNA BINDING ACTIVITY THROUGH THE N-TERMINAL REGION OF THE PROTEIN.
Dose amountVAR
Number1
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionDOSE