Experiment 519168

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationDERRY,WB: WILSON,L: JORAN,MA:. (1995). SUBSTIOCHIOMETRIC BINDING OF TAXOL SUPPRESSES MICROTUBULE DYNAMICS.. 34(7)
Amount utilized
Compound isolated
DiseaseCMPD BINDS TUBULIN AND INHIBITS DISSOCIATIVE ABIILITY. AT CONC <100 NANOMOLAR, SHORTENING OF MICROTUBULE AT PLUS END IS DECREASED. AT CONC <1.0 MICROMULAR, INHIBITS LENGTHENING AND SHORTENING AT BOTH ENDS. AT CONC. >1.0 MICROMOLAR, DYNAMICS ENTIRELY SUPPRESSED.
Dose amountVAR
Number1
Qualitative resultACTIVE
Dose expressionCONC USED