Experiment 520804

Details

PropertyValue
Pharmacology
Administration routeORAL
OrganismCitrus paradisi (RUTACEAE)
CitationHOLLANDER,AAMJ: VAN ROOIJ,J: LENTJES,EWM: ARBOUW,F: VAN BREE,JB: SCHOEMAKER,RC: VAN ES,LA: VAN DER WOUDE,FJ: COHEN,AF:. (1995). THE EFFECT OF GRAPEFRUIT JUICE ON CYCLOSPORINE AND PREDNISONE METABOLISM IN TRANSPLANT PATIENTS.. 57(3)
Amount utilized
Compound isolated
DiseasePLACEBO-CONTROLLED, CROSSOVER STUDY ON EFFECT OF JUICE ON PHARMACOKINETICS OF CYCLOSPORIN IN 12 RENAL TRANSPLANT PATIENTS. JUICE INHIBITS METABOLISM OF CYCLOSPORIN, INCREASING PEAKS. DOES NOT AFFECT AREA UNDER CURVE. DOSED EVERY 3 HOURS X 10.
Dose amount150.0 ML
Number1
Qualitative resultACTIVE
AnimalHUMAN ADULT
Per unitPERSON
Dose expressionDOSE
ExtractJUICE