Experiment 521882

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationLAM,K: CARPENTER,CL: RUDERMAN,NB: FRIEL,JC: KELLY,KL:. (1994). THE PHOSPHATIDYLINOSITOL 3-KINASE SERINE KINASE PHOSPHORYLATES IRS-1.. 269(32)
Amount utilized
Compound isolated
DiseaseBOTH SERINE AND LIPID KINASE ACTIVITIES OF GIVEN ENZYME WERE INHIBITED. ENZYME PHOSPHORYLATES INSULIN RECEPTOR SUBSTRATE-1 IN PRESENCE OF INSULIN, AN EFFECT INHIBITED BY COMPOUND.
Dose amount100.0 NANOMOLS
Number1
Qualitative resultACTIVE
AnimalRAT
Dose expressionCONC USED