Experiment 523526

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationWANG,G: LEMOS,JR:. (1995). TETRANDRINE: A NEW LIGAND TO BLOCK VOLTAGE-DEPENDENT CA2+ AND CA2+-ACTIVATED K+ CHANNELS.. 56(5)
Amount utilized
Compound isolated
DiseaseBLOCKS VOLTAGE-ACTIVATED L-TYPE CHANNELS. CMPD INHIBITS (COMPETITIVELY) DILTIAZEM BINDING, PARTIALLY PREVENTS VERAPAMIL BINDING AND ENHANCES NITRENDIPINE BINDS.
Dose amount4.0 MICROMOLS
Number2
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionIC50