Experiment 524175

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationBERGENDORFF,O: ANKE,H: DEKERMEDJIAN,K: NIELSEN,M: RUDONG,S: STERNER,O: WITT,R:. (1994). THE AFFINITY OF CYCLODEPSIPEPTIDES TO THE BRAIN CHLORIDE CHANNEL DOMAIN OF THE GABAA RECEPTOR IN VITRO.. 47(12)
Amount utilized
Compound isolated
DiseaseCMPD DISPLACES LABELED TERT-BUTYLBICYCLO PHOSPHOROTHIOHNATE FROM GABA-A-RECEPTOR-ASSOCIATED CHLORIDE CHANNEL.
Dose amount16.0 MCG
Number1
Qualitative resultACTIVE
AnimalRAT
Per unitML
Dose expressionIC50