Experiment 526238
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | HARDICK,DJ: COOPER,G: SCOTT-WARD,T: BLAGBROUGH,IS: POTTER,BVL: WONNACOTT,S:. (1995). CONVERSION OF THE SODIUM CHANNEL ACTIVATOR ACONITINE INTO A POTENT ALPHA-7-SELECTIVE NICOTINIC LIGAND.. 365(1) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND HAS PREFERENTIAL AFFINITY FOR ALPHA-BUNGAROTOXIN-BINDING RECEPTORS, BUT MUCH LESS THAN THAT OF PARENT COMPOUND, METHYLLYCACONITINE. |
| Dose amount | 10.0 MG |
| Number | 6 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Dose expression | CONC USED |