Experiment 535829

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationBOWEN,WD: VILNER,BJ: WILLIAMS,W: BERTHA,CM: KUEHNE,ME: JACOBSON,AE:. (1995). IBOGAINE AND ITS CONGENERS ARE DELTA2 RECEPTOR-SELECTIVE LIGANDS WITH MODERATE AFFINITY.. 279(1)
Amount utilized
Compound isolated
DiseaseCMPD BINDS TO SIGMA-2 OPIOID RECEPTOR WITH LESSER AFFINITY THAN TO SIGMA-1 RECEPTOR.
Dose amount19.8 MICROMOLS
Number6
Qualitative resultWEAK ACTIVITY
AnimalGUINEA PIG
Dose expressionCONC USED