Experiment 537399

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationMARKOVITS,J: JUNOLIA,S: COLDWASSER,F: VENUAT,AM: LUCCIONI,C: BEAUMATIN,J: SAUCER,JM: BERNIHEIM,A: JACQUEMIN-SABLON,A:. (1995). GENISTEIN RESISTANCE IN HUMAN LEUKAEMIC CCRF-CEM CELLS: SELECTION OF A DIPLOID CELL LINE WITH REDUCED DNA TOPOISOMERASE II BETA ISOFORM.. 50(2)
Amount utilized
Compound isolated
DiseaseMECHANISTIC STUDY: RESISTANT STRAINS HAD A REDUCED EXPRESSION OF TOPOISOMERASE II BETA ISOFORM WHICH CONFIRMS THAT GENISTEIN'S CYTOTOXICITY IS RELATED TO TOPOISOMERASE II INHIBITION.
Dose amount20.0 MICROMOLS
Number1
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionIC50