Experiment 547976
Worktypes
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | ORAL |
| Organism | Citrus paradisi (RUTACEAE) |
| Citation | LUNDAHL,J: REGARDH,CG: EDGAR,B: JOHNSSON,G:. (1995). RELATIONSHIP BETWEEN TIME OF INTAKE OF GRAPEFRUIT JUICE AND ITS EFFECT ON PHARMACOKINETICS AND PHARMACODYNAMICS OF FELODIPINE IN HEALTHY SUBJECTS.. 49(1/2) |
| Amount utilized | |
| Compound isolated | |
| Disease | EXTRACT INCREASED MAXIMUM SERUM CONCENTRATIONS AND AREA-UNDER-CURVE FOR FELODIPINE IN NINE HEALTHY VOLUNTEERS IN RANDOMIZED, CROSS-OVER STUDY. EXTRACT APPEARS TO INHIBIT FELODIPINE METABOLISM UP TO 24 HOURS POST INGESTION OF JUICE. |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |
| Extract | JUICE |