Experiment 548467

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationFALYNEK,CR: SCHROEDER,J: MAUVAIS,P: MILLER,D: WANG,S: MURPHY,D: LEHR,R: KELLEY,M: MAYCOCK,A: MICHNE,W: MISKI,M: THUNBERG,AL:. (1995). DAMNACANTHAL IS A HIGHLY POTENT, SELECTIVE INHIBITOR OF P56LCK TYROSINE KINASE ACTIVITY.. 34(38)
Amount utilized
Compound isolated
DiseaseWAS SELECTIVE INHIBITOR OF P56-LCK ENZYME, BUT WAS NOT ACTIVE IN WHOLE CELL ASSAYS.
Dose amount0.62 MICROMOLS
Number1
Qualitative resultACTIVE
Dose expressionIC50