Experiment 552600
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | SLEPNEVA,IA: SERGEEVA,SV: KHRAMTSOV,VV:. (1995). REVERSIBLE INHIBITION OF NADPH-CYTOCHROME P450 REDUCTASE BY ALPHA-LIPOIC ACID.. 214(3) |
| Amount utilized | |
| Compound isolated | |
| Disease | NADP COMPLETELY PROTECTED REDUCTASE FROM THE INACTIVATION. THE MODIFICATION OF REDUCTASE WAS REVERSIBLE. THE MODIFIED ENZYME WAS PARTIALLY REACTIVATED WITH DITHIOTHREITOL AND DIHYDROLIPOIC ACID IN THE CASE WHEN CYTOCHROME C WAS A SUBSTRATE SUBSTRATE OF REDUCTASE. AGENT ALPHA-LIPOIC ACID IS AN EFFICIENT INHIBITOR OF BOTH PURIFIED AND MICROSAOMAL REDUCTASE. |
| Dose amount | 0.1 MILLIMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Dose expression | CONC USED |