Experiment 560370

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationDUMONTET,C: DURAN,GE: STEGER,KA: BEKETIC-ORESKOVIC,L: SIKIC,BI:. (1996). RESISTANCE MECHANISMS IN HUMAN SARCOMA MUTANTS DERIVED BY SINGLE-STEP EXPOSURE TO PACLITAXEL(TAXOL).. 56(5)
Amount utilized
Compound isolated
DiseaseEXPOSURE TO CMPD RESULTED IN RESISTANT CLONES ONLY HALF OF WHICH EXPRESSED MDR-1 GENE BUT ALL OF WHICH HAD REDUCED EXPRESSION OF BETA-4 AND 5-BETA TUBULIN ISOTYPES.
Dose amount10.0
Number1
Qualitative resultACTIVE
AnimalCELL CULTURE
Dose expressionCONC USED