Experiment 565728

Details

PropertyValue
Pharmacology
OrganismMaprounea africana (EUPHORBIACEAE)
CitationPENGSUPARP,T: CAI,L: CONSTANT,H: FONG,HHS: LIN,LZ: KINGHORN,AD: PEZZUTO,JM: CORDELL,GA: INGOLFSDOTTIR,K: WAGNER,H: HUGHES,SH:. (1995). MECHANISTIC EVALUATION OF NEW PLANT-DERIVED COMPOUNDS THAT INHIBIT HIV-1 REVERSE TRANSCRIPTASE.. 58(7)
Amount utilized
Compound isolated
DiseaseINHIBITION INVOLVES NON-SPECIFIC BINDING TO THE ENZYME AT NON SUBSTRATE BINDING SITES.
Dose amount15.1 MICROMOLS
Number4
Qualitative resultACTIVE
Dose expressionIC50