Experiment 583860
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | GOLDWASSER,F: SHIMIZU,T: JACKMAN,J: HOKI,Y: O'CONNER,PM: KOHN,KW: POMMIER,Y:. (1996). CORRELATIONS BETWEEN S AND G2 ARREST AND THE CYTOTOXICITY OF CAMPTOTHECIN IN HUMAN COLON CARCINOMA CELLS.. 56(19) |
| Amount utilized | |
| Compound isolated | |
| Disease | COMPOUND APPEARS TO HAVE TWO CYTOTOXIC MECHANISMS, ONE ASSOCIATED WITH DEFICIENCY IN DAMAGED REPLICON ELONGATION AND GREATER CAPACITY TO BREAK THROUGH G2 CHECKPOINT AFTER DNA DAMAGE. THESE ATTRIBUTES CORRELATE WITH SENSITIVITY TO THE COMPOUND. |
| Dose amount | 0.5 MICROMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | IC90 |