Experiment 607457
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | EXTERNAL |
| Organism | Empty organism |
| Citation | AHLUWALIA,GS: SHANDER,D: STYCZYNSKI,P:. (1996). INHIBITION OF HAIR GROWTH WITH PROTEIN KINASE C INHIBITORS.. () |
| Amount utilized | |
| Compound isolated | |
| Disease | MAMMALIAN HAIR GROWTH IS REDUCED BY APPLYING TO THE SKIN A COMPN. INCLUDING AN INHIBITOR OF PROTEIN KINASE C (PKC). THE INHIBITOR INTERACTS WITH THE ATP-BINDING SITE, CA-BINDING SITE, OR PHOSPHOLIPID->30% WHEN TESTED IN THE GOLDEN SYRIAN HAMSTER ASSAY. A NO. OF PKC INHIBITORS WERE TESTED IN THE GOLDEN SYRIAN HAMSTER ASSAY; E.G. VERAPAMIL, THIORIDAZINE, CURCUMIN, AND TRIFLUOPERAZINE INHIBITED HAIR GROWTH BY 56-69%. |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | HAMSTER |
| Dose expression | CONC USED |